Compile Data Set for Download or QSAR
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Found 3 Enz. Inhib. hit(s) with Target = 'Tyrosine-protein kinase SRC' and Monomerid = 50074242
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Aventis

Curated by ChEMBL
LigandPNGBDBM50074242((2S,3S)-2-((S)-2-{(S)-2-[(S)-2-Acetylamino-3-(4-ph...)
Affinity DataIC50:  9nMAssay Description:Binding affinity for Src SH2 domain in scintillation proximity binding assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Aventis

Curated by ChEMBL
LigandPNGBDBM50074242((2S,3S)-2-((S)-2-{(S)-2-[(S)-2-Acetylamino-3-(4-ph...)
Affinity DataIC50:  150nMAssay Description:Binding affinity for p60 c-Src SH2 domain by scintillation proximity assay (SPA)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProto-oncogene tyrosine-protein kinase Src(Homo sapiens (Human))
Aventis

Curated by ChEMBL
LigandPNGBDBM50074242((2S,3S)-2-((S)-2-{(S)-2-[(S)-2-Acetylamino-3-(4-ph...)
Affinity DataIC50:  6.50E+3nMAssay Description:Concentration of compoound required for inhibiting the binding of the fluorescent probe to the c-Src tyrosine kinase SH2 domain by 50%More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed