BindingDB PrimarySearch

Found 2 hits Enz. Inhib. hit(s) with Target = 'Retinoic acid receptor alpha' and Monomerid = 50075880
Target/Host (Institution)	Ligand	Target/Host Links	Ligand Links	Trg + Lig Links	Ki nM	ΔG° kJ/mole	IC50 nM	Kd nM	EC50/IC50 nM	k_off s^-1	k_on M^-1s^-1	pH	Temp °C
Retinoid X receptor gamma/retinoic acid receptor alpha (Homo sapiens (Human))	BDBM50075880 (4-(5,5-Dimethyl-8-p-tolyl-5,6-dihydro-anthracen-2-...) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt UniProtKB/TrEMBL B.MOAD DrugBank antibodypedia GoogleScholar	CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	20	n/a	n/a	n/a	n/a	n/a	n/a
Allergan Inc Curated by ChEMBL					Assay Description Antagonistic activity against RAR alpha in transcriptional activation assay with 32 nM TTNPB				Bioorg Med Chem Lett 9: 743-8 (1999) Article DOI: 10.1016/s0960-894x(99)00077-3 BindingDB Entry DOI: 10.7270/Q26Q1WFP
Allergan Inc Curated by ChEMBL					More data for this Ligand-Target Pair
Retinoic acid receptor alpha/Retinoid X receptor alpha (Homo sapiens (Human))	BDBM50075880 (4-(5,5-Dimethyl-8-p-tolyl-5,6-dihydro-anthracen-2-...) Show SMILES Show InChI	PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt UniProtKB/TrEMBL B.MOAD DrugBank antibodypedia GoogleScholar	CHEMBL PC cid PC sid UniChem	Article PubMed	n/a	n/a	n/a	13	n/a	n/a	n/a	n/a	n/a
Allergan Inc Curated by ChEMBL					Assay Description Antagonistic activity against RAR alpha in transcriptional activation assay with 32 nM TTNPB				Bioorg Med Chem Lett 9: 743-8 (1999) Article DOI: 10.1016/s0960-894x(99)00077-3 BindingDB Entry DOI: 10.7270/Q26Q1WFP
Allergan Inc Curated by ChEMBL					More data for this Ligand-Target Pair