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Found 1 hit Enz. Inhib. hit(s) with Target = 'Telomerase reverse transcriptase' and Monomerid = 50082532   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Telomerase reverse transcriptase


(Homo sapiens (Human))
BDBM50082532
PNG
(2,6-Bis(3-piperidinopropionamido)anthracene-9,10-d...)
Show SMILES Oc1c2ccc(NC(=O)CC[NH+]3CCCCC3)cc2c(O)c2ccc(NC(=O)CC[NH+]3CCCCC3)cc12
Show InChI InChI=1S/C30H38N4O4/c35-27(11-17-33-13-3-1-4-14-33)31-21-7-9-23-25(19-21)29(37)24-10-8-22(20-26(24)30(23)38)32-28(36)12-18-34-15-5-2-6-16-34/h7-10,19-20,37-38H,1-6,11-18H2,(H,31,35)(H,32,36)/p+2
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Similars

Article
PubMed
n/an/a 4.50E+3n/an/an/an/an/an/a



The Institute of Cancer Research

Curated by ChEMBL


Assay Description
Inhibitory activity against Telomerase evaluated by TRAP Assay studies.


J Med Chem 42: 4538-46 (1999)


Article DOI: 10.1021/jm990287e
BindingDB Entry DOI: 10.7270/Q2J103VC
More data for this
Ligand-Target Pair