Compile Data Set for Download or QSAR
maximum 50k data
Found 3 Enz. Inhib. hit(s) with Target = 'Adenosine Receptor A1' and Monomerid = 50086146
TargetAdenosine receptor A1(BOVINE)
Universita' Di Firenze

Curated by ChEMBL
LigandPNGBDBM50086146(CHEMBL16305 | N-(1-Oxo-2-phenyl-1,2-dihydro-[1,2,4...)
Affinity DataKi:  4.30nMAssay Description:Binding affinity towards adenosine A1 receptor of bovine brain membrane in presence of [3H]-CHA at a concentration of 20 uMMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(BOVINE)
Universita' Di Firenze

Curated by ChEMBL
LigandPNGBDBM50086146(CHEMBL16305 | N-(1-Oxo-2-phenyl-1,2-dihydro-[1,2,4...)
Affinity DataKi:  4.30nMAssay Description:Displacement of [3H]DPCPX from adenosine A1 receptor in bovine brain membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Università

Curated by ChEMBL
LigandPNGBDBM50086146(CHEMBL16305 | N-(1-Oxo-2-phenyl-1,2-dihydro-[1,2,4...)
Affinity DataKi:  2.00E+3nMAssay Description:Displacement of [3H]DPCPX from human adenosine A1 receptor expressed in CHO cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed