Affinity DataKi: 5.02nMAssay Description:Antagonist activity against adenosine A1 receptor in rat brain membrane in presence of [3H]-R-PIA radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 54.7nMAssay Description:Antagonist activity against recombinant human adenosine A1 receptor expressed in HEK-293 cells in presence of [125I]-IABA radioligand.More data for this Ligand-Target Pair
Affinity DataKi: 63.1nMAssay Description:Binding affinity to recombinant human adenosine A1 receptorMore data for this Ligand-Target Pair