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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Excitatory amino acid transporter 1' and Monomerid = 50088220   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Excitatory amino acid transporter 1


(Homo sapiens (Human))
BDBM50088220
PNG
((2S,4R)-4-pentylglutamic acid | 2-Amino-4-pentyl-p...)
Show SMILES CCCCC[C@H](C[C@H](N)C(O)=O)C(O)=O
Show InChI InChI=1S/C10H19NO4/c1-2-3-4-5-7(9(12)13)6-8(11)10(14)15/h7-8H,2-6,11H2,1H3,(H,12,13)(H,14,15)/t7-,8+/m1/s1
Reactome pathway
KEGG

UniProtKB/SwissProt

DrugBank
GoogleScholar
CHEMBL
PC cid
PC sid
UniChem

Similars

Article
PubMed
1.20E+5n/an/an/an/an/an/an/an/a



Université Blaise Pascal

Curated by ChEMBL


Assay Description
Binding affinity to human EAAT1 expressed in HEK293 cells in FMP (FLPR) assay


J Med Chem 48: 7980-92 (2005)


Article DOI: 10.1021/jm050597z
BindingDB Entry DOI: 10.7270/Q2MP52V1
More data for this
Ligand-Target Pair