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Found 2 Enz. Inhib. hit(s) with Target = 'Alpha-1a adrenergic receptor' and Monomerid = 50088706
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50088706(CHEMBL12062 | N-{3-[4-(2-Isopropoxy-phenyl)-pipera...)
Affinity DataKi:  0.650nMAssay Description:Binding constant measured against Alpha-1A adrenergic receptor in human prostate; +++:highly activeMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-1A adrenergic receptor(Homo sapiens (Human))
China Pharmaceutical University

Curated by ChEMBL
LigandPNGBDBM50088706(CHEMBL12062 | N-{3-[4-(2-Isopropoxy-phenyl)-pipera...)
Affinity DataKi:  0.660nMAssay Description:Binding affinity for human Alpha-1A adrenergic receptor expressed in COS cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed