Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with Target = 'Adenosine Receptor A1' and Monomerid = 50100417
TargetAdenosine receptor A1(Rattus norvegicus (rat))
Niddk

Curated by ChEMBL
LigandPNGBDBM50100417((1R,2S,4S,5S)-4-(2-Chloro-6-cyclopentylamino-purin...)
Affinity DataKi:  3.60E+3nMAssay Description:Ability to displace specific radioligand [3H]R-PIA binding at Adenosine A1 receptor in rat brain membraneMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A1(Homo sapiens (Human))
Niddk

Curated by ChEMBL
LigandPNGBDBM50100417((1R,2S,4S,5S)-4-(2-Chloro-6-cyclopentylamino-purin...)
Affinity DataEC50:  2.28E+3nMAssay Description:Agonist efficacy as effective concentration to stimulate binding of [35S]GTP-gamma-S, at human Adenosine A1 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed