Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Urokinase-type plasminogen activator (Homo sapiens (Human)) | BDBM50102777![]() (2-(5-Fluoro-2-hydroxy-phenyl)-1H-benzoimidazole-5-...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt UniProtKB/TrEMBL B.MOAD DrugBank antibodypedia GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.80E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Axys Pharmaceuticals Inc Curated by ChEMBL | Assay Description ComInhibition of Human Serine Protease Urokinase Plasminogen Activator (u-PA). | J Med Chem 44: 2753-71 (2001) Article DOI: 10.1021/jm0100638 BindingDB Entry DOI: 10.7270/Q2RX9BC7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Plasminogen (Homo sapiens (Human)) | BDBM50102777![]() (2-(5-Fluoro-2-hydroxy-phenyl)-1H-benzoimidazole-5-...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 2.10E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Axys Pharmaceuticals Inc Curated by ChEMBL | Assay Description Inhibition of Human Serine Protease Plasmin. | J Med Chem 44: 2753-71 (2001) Article DOI: 10.1021/jm0100638 BindingDB Entry DOI: 10.7270/Q2RX9BC7 | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Tissue-type plasminogen activator (Homo sapiens (Human)) | BDBM50102777![]() (2-(5-Fluoro-2-hydroxy-phenyl)-1H-benzoimidazole-5-...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt B.MOAD DrugBank antibodypedia GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 4.60E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Axys Pharmaceuticals Inc Curated by ChEMBL | Assay Description Inhibition of Human Serine Protease tissue type Plasminogen Activator (t-PA). | J Med Chem 44: 2753-71 (2001) Article DOI: 10.1021/jm0100638 BindingDB Entry DOI: 10.7270/Q2RX9BC7 | |||||||||||
More data for this Ligand-Target Pair |