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Found 2 Enz. Inhib. hit(s) with Target = 'Glucagon receptor' and Monomerid = 50104369
TargetGlucagon receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50104369(4-[5-(4-Fluoro-phenyl)-2-naphthalen-1-yl-3H-imidaz...)
Affinity DataIC50:  340nMAssay Description:Inhibition of human glucagon receptor expressed in CHO cell membranes by radioligand displacement assayMore data for this Ligand-Target Pair
In DepthDetails Article
TargetGlucagon receptor(Homo sapiens (Human))TBA
LigandPNGBDBM50104369(4-[5-(4-Fluoro-phenyl)-2-naphthalen-1-yl-3H-imidaz...)
Affinity DataIC50:  1.50E+3nMAssay Description:Binding affinity towards human glucagon receptor in absence of Mg2+ expressed as IC50More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed