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Found 2 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M1' and Monomerid = 50107709
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
The University Of Toledo

Curated by ChEMBL
LigandPNGBDBM50107709(1,11-di[4-(1-methyl-1,2,3,6-tetrahydro-5-pyridinyl...)
Affinity DataKi:  0.570nMAssay Description:Binding affinity towards M1 muscarinic receptor expressed in A9 L cells by diaplacing [3H]-(R)-QNB radioligand.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMuscarinic acetylcholine receptor M1(Homo sapiens (Human))
The University Of Toledo

Curated by ChEMBL
LigandPNGBDBM50107709(1,11-di[4-(1-methyl-1,2,3,6-tetrahydro-5-pyridinyl...)
Affinity DataEC50:  1.50E+3nMAssay Description:Agonistic activity against M1 muscarinic receptor expressed in A9 L cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed