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Compile Data Set for Download or QSAR

Found 1 hit Enz. Inhib. hit(s) with Target = 'Excitatory amino acid transporter 1' and Monomerid = 50107948   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Excitatory amino acid transporter 1


(Homo sapiens (Human))
BDBM50107948
PNG
(2-Amino-3-(2-hydroxy-2H-pyrazol-3-yl)-propionic ac...)
Show SMILES NC(Cc1ccnn1O)C(O)=O
Show InChI InChI=1/C6H9N3O3/c7-5(6(10)11)3-4-1-2-8-9(4)12/h1-2,5,12H,3,7H2,(H,10,11)
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CHEMBL
PC cid
PC sid
UniChem

Similars

Article
PubMed
n/an/a>1.00E+6n/an/an/an/an/an/a



The Royal Danish School of Pharmacy

Curated by ChEMBL


Assay Description
Binding affinity for Excitatory amino acid transporter 1 (EAAT-1) in Glu uptake system


J Med Chem 45: 19-31 (2001)


Article DOI: 10.1021/jm010303j
BindingDB Entry DOI: 10.7270/Q2KH0MMK
More data for this
Ligand-Target Pair