Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Adenosine Receptor A2A' and Monomerid = 50108039
TargetAdenosine receptor A2a(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50108039(4-(3-(5-amino-2-(furan-2-yl)-7H-pyrazolo[4,3-e][1,...)
Affinity DataKi:  140nMAssay Description:Displacement of [3H]NECA from human adenosine A2A receptor expressed in CHO cellsChecked by AuthorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50108039(4-(3-(5-amino-2-(furan-2-yl)-7H-pyrazolo[4,3-e][1,...)
Affinity DataKi:  140nMAssay Description:Displacement of [3H]-SCH- 58261 binding at human Adenosine A2A receptor expressed in HEK-293 cells; ranges from 129-152More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed