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Found 1 hit Enz. Inhib. hit(s) with Target = 'Telomerase reverse transcriptase' and Monomerid = 50108801   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Telomerase reverse transcriptase


(Homo sapiens (Human))
BDBM50108801
PNG
(6,8,13-trimethyl-8H-quino[4,3,2-kl]acridin-13-ium;...)
Show SMILES Cc1cc2n(C)c3ccccc3c3[n+](C)c4ccccc4c(c1)c23
Show InChI InChI=1S/C22H19N2/c1-14-12-17-15-8-4-6-10-18(15)24(3)22-16-9-5-7-11-19(16)23(2)20(13-14)21(17)22/h4-13H,1-3H3/q+1
PDB

NCI pathway
Reactome pathway
KEGG

UniProtKB/SwissProt

DrugBank
antibodypedia
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CHEMBL
PC cid
PC sid
UniChem

Similars

Article
PubMed
n/an/a 760n/an/an/an/an/an/a



University of Nottingham

Curated by ChEMBL


Assay Description
Inhibition of telomerase activity using TRAP assay


J Med Chem 45: 590-7 (2002)


Article DOI: 10.1021/jm011015q
BindingDB Entry DOI: 10.7270/Q2BR8RGQ
More data for this
Ligand-Target Pair