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Found 2 Enz. Inhib. hit(s) with Target = 'Telomerase reverse transcriptase' and Monomerid = 50108802
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50108802(3,11-difluoro-6,8,13-trimethyl-8H-quino[4,3,2-kl]a...)
Affinity DataIC50:  330nMAssay Description:Inhibition of telomerase activity using TRAP assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTelomerase reverse transcriptase(Homo sapiens (Human))
University Of Nottingham

Curated by ChEMBL
LigandPNGBDBM50108802(3,11-difluoro-6,8,13-trimethyl-8H-quino[4,3,2-kl]a...)
Affinity DataIC50:  3.31E+8nMAssay Description:Inhibition of Homo sapiens (human) telomerase assessed as formation of G-tetraplexes by gel mobility shift assayMore data for this Ligand-Target Pair
In DepthDetails Article