Compile Data Set for Download or QSAR
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Found 4 Enz. Inhib. hit(s) with Target = 'Peroxisome proliferator-activated receptor alpha' and Monomerid = 50109554
LigandPNGBDBM50109554(3-{4-[2-(3,6-Dibromo-carbazol-9-yl)-ethoxy]-phenyl...)
Affinity DataEC50:  220nMAssay Description:Transactivation of GAL4-fused Homo sapiens (human) PPARalpha DNA binding domain expressed in African green monkey CV1 cells by luciferase reporter ge...More data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50109554(3-{4-[2-(3,6-Dibromo-carbazol-9-yl)-ethoxy]-phenyl...)
Affinity DataEC50:  219nMAssay Description:Transactivation of Homo sapiens (human) PPARalpha assessed as luciferase activity by reporter gene assayMore data for this Ligand-Target Pair
In DepthDetails Article
LigandPNGBDBM50109554(3-{4-[2-(3,6-Dibromo-carbazol-9-yl)-ethoxy]-phenyl...)
Affinity DataEC50:  220nMAssay Description:In vitro transactivation using receptor transactivation assay against hPPAR alphaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
LigandPNGBDBM50109554(3-{4-[2-(3,6-Dibromo-carbazol-9-yl)-ethoxy]-phenyl...)
Affinity DataEC50:  220nMAssay Description:Transactivation of GAL4-fused Homo sapiens (human) PPARalpha DNA binding domain expressed in African green monkey CV1 cells by luciferase reporter ge...More data for this Ligand-Target Pair
In DepthDetails Article