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Found 2 Enz. Inhib. hit(s) with Target = 'Tyrosine-protein kinase LCK' and Monomerid = 50112928
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
University Of Zurich

Curated by ChEMBL
LigandPNGBDBM50112928((2-Bromo-phenyl)-(3-phenyl-imidazo[1,5-a]quinoxali...)
Affinity DataIC50: >1.25E+4nMAssay Description:Inhibition of LckMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetTyrosine-protein kinase Lck(Homo sapiens (Human))
University Of Zurich

Curated by ChEMBL
LigandPNGBDBM50112928((2-Bromo-phenyl)-(3-phenyl-imidazo[1,5-a]quinoxali...)
Affinity DataIC50: >1.25E+4nMAssay Description:Inhibitory activity against recombinant p56 Lck tyrosine kinase expressed as a His-tagged protein in insect cells using a baculovirus expression syst...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed