Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Urokinase-type plasminogen activator (Homo sapiens (Human)) | BDBM50115897![]() (CHEMBL64841 | N-(4-Guanidino-phenyl)-2-hydroxy-5-m...) | PDB MMDB Reactome pathway KEGG UniProtKB/SwissProt UniProtKB/TrEMBL B.MOAD DrugBank antibodypedia GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 1.30E+4 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Celera Curated by ChEMBL | Assay Description Inhibition of urokinase-type plasminogen activator (microPa) | Bioorg Med Chem Lett 12: 2023-6 (2002) Article DOI: 10.1016/s0960-894x(02)00312-8 BindingDB Entry DOI: 10.7270/Q2ZG6RK4 | |||||||||||
More data for this Ligand-Target Pair |