Found 2 Enz. Inhib. hit(s) with Target = 'Peroxisome Proliferator-Activated Receptor gamma' and Monomerid = 50121412
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Biovitrum
Curated by ChEMBL
Biovitrum
Curated by ChEMBL
Affinity DataKi: 2.20E+3nMAssay Description:Ligand binding affinity was determined by displacement of a tritiated tracer by the unlabeled compound to a GST-PPAR fusion protein for Peroxisome pr...More data for this Ligand-Target Pair
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Biovitrum
Curated by ChEMBL
Biovitrum
Curated by ChEMBL
Affinity DataEC50: 1.60E+3nMAssay Description:Transactivation potency was measured by luciferase activity in Caco- 2/TC7 cells transiently co-transfected for the fusion-protein Gal4-PPAR gammaMore data for this Ligand-Target Pair