Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Peroxisome Proliferator-Activated Receptor gamma' and Monomerid = 50121424
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Biovitrum

Curated by ChEMBL
LigandPNGBDBM50121424(CHEMBL119111 | Lithium; 5-(6-chloro-pyrazin-2-ylox...)
Affinity DataKi:  160nMAssay Description:Ligand binding affinity was determined by displacement of a tritiated tracer by the unlabeled compound to a GST-PPAR fusion protein for Peroxisome pr...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Biovitrum

Curated by ChEMBL
LigandPNGBDBM50121424(CHEMBL119111 | Lithium; 5-(6-chloro-pyrazin-2-ylox...)
Affinity DataEC50:  450nMAssay Description:Transactivation potency was measured by luciferase activity in Caco- 2/TC7 cells transiently co-transfected for the fusion-protein Gal4-PPAR gammaMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed