Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with Target = 'Peroxisome Proliferator-Activated Receptor gamma' and Monomerid = 50124382
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50124382(3-Methyl-3-{4-[4-(3-phenyl-7-propyl-benzo[d]isoxaz...)
Affinity DataKi:  52nMAssay Description:In vitro binding affinity towards human peroxisome proliferator activated receptor gamma (PPAR gamma)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor gamma(Homo sapiens (Human))
Merck Research Laboratories

Curated by ChEMBL
LigandPNGBDBM50124382(3-Methyl-3-{4-[4-(3-phenyl-7-propyl-benzo[d]isoxaz...)
Affinity DataEC50:  37nMAssay Description:Agonistic activity was determined in COS1 cells transfected with GAL 4-PPAR alpha receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed