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Found 4 Enz. Inhib. hit(s) with Target = 'Nischarin' and Monomerid = 50127572
TargetNischarin(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50127572(2-(4,5-Dihydro-1H-imidazol-2-yl)-6-fluoro-4-methyl...)
Affinity DataKi:  17nMAssay Description:In vitro binding affinity determined against imidazoline receptor I-2 using rabbit kidney preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50127572(2-(4,5-Dihydro-1H-imidazol-2-yl)-6-fluoro-4-methyl...)
Affinity DataKi:  31nMAssay Description:In vitro binding affinity determined against imidazoline receptor I-1 from rabbit kidney preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50127572(2-(4,5-Dihydro-1H-imidazol-2-yl)-6-fluoro-4-methyl...)
Affinity DataKi:  31nMAssay Description:In vitro binding affinity determined against imidazoline receptor I-1 from rabbit kidney preparationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetNischarin(Homo sapiens (Human))
Université

Curated by ChEMBL
LigandPNGBDBM50127572(2-(4,5-Dihydro-1H-imidazol-2-yl)-6-fluoro-4-methyl...)
Affinity DataKi:  63nMAssay Description:Binding affinity for imidazoline receptor I-2 in rabbit kidney homogenate (relative to [3H]-Idazoxan radioligand)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed