Compile Data Set for Download or QSAR
maximum 50k data
Found 4 Enz. Inhib. hit(s) with Target = 'Progesterone receptor' and Monomerid = 50129171
TargetProgesterone receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50129171(9-Bromo-7-fluoro-2,2,4-trimethyl-2,5-dihydro-1H-6-...)
Affinity DataKi:  12nMAssay Description:Binding affinity at human progesterone receptor.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50129171(9-Bromo-7-fluoro-2,2,4-trimethyl-2,5-dihydro-1H-6-...)
Affinity DataKi:  12nMAssay Description:Displacement of [3H]progesterone from Progesterone receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50129171(9-Bromo-7-fluoro-2,2,4-trimethyl-2,5-dihydro-1H-6-...)
Affinity DataIC50:  461nMAssay Description:Inhibition of human progesterone receptor activation in T47D human breast cancer cell.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Ligand Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50129171(9-Bromo-7-fluoro-2,2,4-trimethyl-2,5-dihydro-1H-6-...)
Affinity DataEC50:  57nMAssay Description:Antagonistic activity at human progesterone receptor in CV-1 cells.More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed