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Found 2 Enz. Inhib. hit(s) with Target = 'Prolyl endopeptidase' and Monomerid = 50134163
TargetProlyl endopeptidase(Sus scrofa)
University Of Kuopio

Curated by ChEMBL
LigandPNGBDBM50134163((S)-1-((S)-1-{3-[(S)-2-(Pyrrolidine-1-carbonyl)-py...)
Affinity DataIC50:  1.5nMpH: 7.0Assay Description:In vitro inhibitory activity against porcine prolyl oligopeptidase by using 4 mM Suc-Gly-Pro-7-amido-4-methylcoumarin as substrate (pH 7.0) at 30 deg...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProlyl endopeptidase(Sus scrofa)
University Of Kuopio

Curated by ChEMBL
LigandPNGBDBM50134163((S)-1-((S)-1-{3-[(S)-2-(Pyrrolidine-1-carbonyl)-py...)
Affinity DataIC50:  1.5nMAssay Description:In vitro inhibition of prolyl oligopeptidase (POP) from pig brainMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed