Target/Host (Institution) | Ligand | Target/Host Links | Ligand Links | Trg + Lig Links | Ki nM | ΔG° kJ/mole | IC50 nM | Kd nM | EC50/IC50 nM | koff s-1 | kon M-1s-1 | pH | Temp °C |
---|---|---|---|---|---|---|---|---|---|---|---|---|---|
Retinoid X receptor gamma/retinoic acid receptor alpha (Homo sapiens (Human)) | BDBM50135463![]() ((2E,4E,6Z)-7-[2-(2,2-Difluoro-ethoxy)-5-isopropyl-...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt UniProtKB/TrEMBL B.MOAD DrugBank antibodypedia GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 23 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Ligand Pharmaceuticals Inc Curated by ChEMBL | Assay Description Binding affinity against RXR gamma receptor using [3H]-9-cis-RA as radioligand in CV-1 cells | Bioorg Med Chem Lett 13: 4071-5 (2003) Article DOI: 10.1016/j.bmcl.2003.08.048 BindingDB Entry DOI: 10.7270/Q2V987GP | |||||||||||
More data for this Ligand-Target Pair | |||||||||||||
Retinoid X receptor gamma/retinoic acid receptor alpha (Homo sapiens (Human)) | BDBM50135463![]() ((2E,4E,6Z)-7-[2-(2,2-Difluoro-ethoxy)-5-isopropyl-...) | PDB MMDB NCI pathway Reactome pathway KEGG UniProtKB/SwissProt UniProtKB/TrEMBL B.MOAD DrugBank antibodypedia GoogleScholar | CHEMBL PC cid PC sid UniChem Similars | Article PubMed | 4.66E+3 | n/a | n/a | n/a | n/a | n/a | n/a | n/a | n/a |
Ligand Pharmaceuticals Inc Curated by ChEMBL | Assay Description Binding affinity against RAR alpha receptor using [3H]-ATRA as radioligand in CV-1 cells | Bioorg Med Chem Lett 13: 4071-5 (2003) Article DOI: 10.1016/j.bmcl.2003.08.048 BindingDB Entry DOI: 10.7270/Q2V987GP | |||||||||||
More data for this Ligand-Target Pair |