Compile Data Set for Download or QSAR
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Found 3 Enz. Inhib. hit(s) with Target = 'Adenosine Receptor A2B' and Monomerid = 50140942
TargetAdenosine receptor A2b(Homo sapiens (Human))
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Curated by ChEMBL
LigandPNGBDBM50140942(CHEMBL33491 | N-(3,4-Dimethyl-phenyl)-2-[5-(2,6-di...)
Affinity DataKi:  10nMAssay Description:Binding affinity of compound for displacement of [3H]DPCPX binding in HEK293 membranes expressing human A2B adenosine receptorsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50140942(CHEMBL33491 | N-(3,4-Dimethyl-phenyl)-2-[5-(2,6-di...)
Affinity DataKi:  10nMAssay Description:Binding affinity of compound for displacement of specific [3H]- DPCPX binding at human A2B receptors expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Universit£

Curated by ChEMBL
LigandPNGBDBM50140942(CHEMBL33491 | N-(3,4-Dimethyl-phenyl)-2-[5-(2,6-di...)
Affinity DataIC50:  40nMAssay Description:Inhibitory activity against cAMP production in CHO cells transfected with human A2B adenosine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed