Compile Data Set for Download or QSAR
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Found 6 Enz. Inhib. hit(s) with Target = 'Glucocorticoid receptor' and Monomerid = 50153512
TargetGlucocorticoid receptor(RAT)
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50153512((9R,10S,11S,13S,14S,16R,17R)-9-Fluoro-11,17-dihydr...)
Affinity DataIC50:  1.40nMAssay Description:Inhibition against U2OS cells expressing rat Glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50153512((9R,10S,11S,13S,14S,16R,17R)-9-Fluoro-11,17-dihydr...)
Affinity DataIC50:  5nMAssay Description:Binding affinity for recombinant human glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50153512((9R,10S,11S,13S,14S,16R,17R)-9-Fluoro-11,17-dihydr...)
Affinity DataEC50:  0.200nMAssay Description:Repression of AP1-luciferase reporter activity in TPA-stimulated U2OS cells expressing rat glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50153512((9R,10S,11S,13S,14S,16R,17R)-9-Fluoro-11,17-dihydr...)
Affinity DataEC50:  5.60nMAssay Description:Effective concentration in CV-1 cell transactivation assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50153512((9R,10S,11S,13S,14S,16R,17R)-9-Fluoro-11,17-dihydr...)
Affinity DataEC50:  0.200nMAssay Description:Effective concentration against MMTV in transactivation assay in U2OS cells expressing rat GRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(RAT)
University Of California San Francisco

Curated by ChEMBL
LigandPNGBDBM50153512((9R,10S,11S,13S,14S,16R,17R)-9-Fluoro-11,17-dihydr...)
Affinity DataEC50:  0.300nMAssay Description:Repression of NFkB-luciferase reporter activity in TPA stimulated U2OS cells expressing rat glucocorticoid receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed