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Found 1 hit Enz. Inhib. hit(s) with Target = 'Telomerase reverse transcriptase' and Monomerid = 50157557   
Target/Host
(Institution)
LigandTarget/Host
Links
Ligand
Links
Trg + Lig
Links
Ki
nM
ΔG°
kJ/mole
IC50
nM
Kd
nM
EC50/IC50
nM
koff
s-1
kon
M-1s-1
pHTemp
°C
Telomerase reverse transcriptase


(Homo sapiens (Human))
BDBM50157557
PNG
(2-(3,4-diaminophenyl)-7,8-dihydroxy-4H-chromen-4-o...)
Show SMILES Nc1ccc(cc1N)-c1cc(=O)c2ccc(O)c(O)c2o1
Show InChI InChI=1S/C15H12N2O4/c16-9-3-1-7(5-10(9)17)13-6-12(19)8-2-4-11(18)14(20)15(8)21-13/h1-6,18,20H,16-17H2
PDB

NCI pathway
Reactome pathway
KEGG

UniProtKB/SwissProt

DrugBank
antibodypedia
GoogleScholar
CHEMBL
PC cid
PC sid
UniChem

Similars

Article
PubMed
n/an/a 3.60E+3n/an/an/an/an/an/a



BU-Nerviano Medical Sciences

Curated by ChEMBL


Assay Description
Inhibition of human telomerase from HEK293 cell extracts by Flash-Plate assay


J Med Chem 47: 6466-75 (2004)


Article DOI: 10.1021/jm040810b
BindingDB Entry DOI: 10.7270/Q2P55N1R
More data for this
Ligand-Target Pair