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Found 2 Enz. Inhib. hit(s) with Target = 'Histamine H3 Receptor' and Monomerid = 50158600
TargetHistamine H3 receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50158600(4-{2-[2-((S)-2-Methyl-pyrrolidin-1-yl)-ethyl]-benz...)
Affinity DataKi:  0.690nMAssay Description:In vitro binding affinity was determined as displacement of [3H]N-R-methylhistamine from C6 cell membranes expressing human histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetHistamine H3 receptor(Rattus norvegicus (rat))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50158600(4-{2-[2-((S)-2-Methyl-pyrrolidin-1-yl)-ethyl]-benz...)
Affinity DataKi:  2.57nMAssay Description:In vitro binding affinity was determined as displacement of [3H]N-R-methylhistamine from C6 cell membranes expressing rat histamine H3 receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed