Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Adenosine Receptor A2A' and Monomerid = 50165066
TargetAdenosine receptor A2a(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50165066(9-Benzyl-6-furan-2-yl-9H-purin-2-ylamine | 9-benzy...)
Affinity DataKi:  34.9nMAssay Description:Inhibition constant against human Adenosine A2a receptor using [3H]-SCH- 58261 as radioligand expressed in HEK cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2a(Homo sapiens (Human))
Schering-Plough Research Institute

Curated by ChEMBL
LigandPNGBDBM50165066(9-Benzyl-6-furan-2-yl-9H-purin-2-ylamine | 9-benzy...)
Affinity DataKi:  40nMAssay Description:Binding affinity at human adenosine A2A receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed