Affinity DataIC50: 4.30nMAssay Description:Inhibition of [125I]-SDF-1 binding to C-X-C chemokine receptor type 4 (CXCR4) expressed in CHO cellsMore data for this Ligand-Target Pair
Affinity DataIC50: 8nMAssay Description:Inhibition of CXCR4 (unknown origin)More data for this Ligand-Target Pair
Affinity DataEC50: 520nMAssay Description:Antagonist activity at human CXCR4 expressed in COS7 cells assessed as inhibition of [3H]inositol-phosphates formation after 90 mins by scintillation...More data for this Ligand-Target Pair
Affinity DataEC50: 525nMAssay Description:Antagonist activity at human CXCR4 expressed in COS7 cells assessed as inhibition of [3H]inositol-phosphates formation after 90 mins by scintillation...More data for this Ligand-Target Pair