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Found 1 Enz. Inhib. hit(s) with Target = 'Alpha-2a adrenergic receptor' and Monomerid = 50170198
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Taisho Pharmaceutical

Curated by ChEMBL
LigandPNGBDBM50170198(CHEMBL362193 | N-[4-(4-Dimethylamino-quinazolin-2-...)
Affinity DataIC50:  130nMAssay Description:Inhibitory activity against alpha-2A adrenergic receptor by using [3H]MK-912 as radioligand expressed in COS-1 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed