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Found 2 Enz. Inhib. hit(s) with Target = 'Glucocorticoid receptor' and Monomerid = 50172040
TargetGlucocorticoid receptor(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50172040(2-Hydroxy-2,4-dimethyl-4-phenyl-pentanoic acid (1-...)
Affinity DataIC50:  370nMAssay Description:Binding affinity towards glucocorticoid receptor using fluorescence polarization competitive binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Boehringer Ingelheim Pharmaceuticals

Curated by ChEMBL
LigandPNGBDBM50172040(2-Hydroxy-2,4-dimethyl-4-phenyl-pentanoic acid (1-...)
Affinity DataEC50:  2.37E+3nMAssay Description:Effective concentration against inhibition of Dexamethasone induced glucocorticoid receptor transactivation of mouse mammary tumor virus luciferase g...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed