Compile Data Set for Download or QSAR
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Found 3 Enz. Inhib. hit(s) with Target = 'Metabotropic glutamate receptor 1' and Monomerid = 50177056
TargetMetabotropic glutamate receptor 1(RAT)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50177056(9-Dimethylamino-3-(2-ethyl-phenyl)-3H-pyrido[3',2'...)
Affinity DataKi:  142nMAssay Description:Displacement of [3H]R214127 from mGluR1 in rat cerebellum membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(RAT)
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50177056(9-Dimethylamino-3-(2-ethyl-phenyl)-3H-pyrido[3',2'...)
Affinity DataIC50:  251nMAssay Description:Inhibition of rat mGluR1More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetMetabotropic glutamate receptor 1(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50177056(9-Dimethylamino-3-(2-ethyl-phenyl)-3H-pyrido[3',2'...)
Affinity DataIC50:  251nMAssay Description:Antagonist activity at human mGluR1 expressed in 1321N1 cells assessed as effect on L-glutamate-induced calcium mobilizationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed