Compile Data Set for Download or QSAR
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Found 3 Enz. Inhib. hit(s) with Target = 'Alpha-2a adrenergic receptor' and Monomerid = 50180251
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50180251(1-((S)-2-aminopropyl)-1H-indazol-6-ol | CHEMBL3713...)
Affinity DataKi:  2.27E+3nMAssay Description:Displacement of [3H]clonidine from cloned human adrenergic alpha2A receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50180251(1-((S)-2-aminopropyl)-1H-indazol-6-ol | CHEMBL3713...)
Affinity DataEC50:  2.60E+3nMAssay Description:Activity at adrenergic alpha2A receptor expressed in human clonic adenocarcinoma HT29 cell by tissue contraction assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAlpha-2A adrenergic receptor(Homo sapiens (Human))
Alcon Research

Curated by ChEMBL
LigandPNGBDBM50180251(1-((S)-2-aminopropyl)-1H-indazol-6-ol | CHEMBL3713...)
Affinity DataEC50: >1.00E+4nMAssay Description:Activity at adrenergic alpha-2A receptor expressed in human clonic adenocarcinoma HT29 cell by adenylyl cyclase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed