Affinity DataKi: 2.27E+3nMAssay Description:Displacement of [3H]clonidine from cloned human adrenergic alpha2A receptor expressed in Sf9 cellsMore data for this Ligand-Target Pair
Affinity DataEC50: 2.60E+3nMAssay Description:Activity at adrenergic alpha2A receptor expressed in human clonic adenocarcinoma HT29 cell by tissue contraction assayMore data for this Ligand-Target Pair
Affinity DataEC50: >1.00E+4nMAssay Description:Activity at adrenergic alpha-2A receptor expressed in human clonic adenocarcinoma HT29 cell by adenylyl cyclase assayMore data for this Ligand-Target Pair