Compile Data Set for Download or QSAR
maximum 50k data
Found 2 Enz. Inhib. hit(s) with Target = 'Peroxisome proliferator-activated receptor alpha' and Monomerid = 50188028
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50188028(2-ethoxy-3-(1-((5-methyl-2-o-tolyloxazol-4-yl)meth...)
Affinity DataIC50:  125nMAssay Description:Binding affinity to PPARalpha by radio ligand binding assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetPeroxisome proliferator-activated receptor alpha(Homo sapiens (Human))
F. Hoffmann-La Roche

Curated by ChEMBL
LigandPNGBDBM50188028(2-ethoxy-3-(1-((5-methyl-2-o-tolyloxazol-4-yl)meth...)
Affinity DataEC50:  830nMAssay Description:Activity at PPARalpha by luciferase reporter gene transactivation assay relative to farglitazarMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed