Found 2 Enz. Inhib. hit(s) with Target = 'Peroxisome Proliferator-Activated Receptor gamma' and Monomerid = 50195080
Affinity DataKi: 300nMAssay Description:Displacement of radiolabeled darglitazone from human PPAR gamma by SPA assayMore data for this Ligand-Target Pair
Affinity DataEC50: 130nMAssay Description:Agonist activity at human PPAR gamma in HepG2 cells by PPAR-GAL4 transactivation assayMore data for this Ligand-Target Pair