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Found 1 Enz. Inhib. hit(s) with Target = 'Metabotropic glutamate receptor 1' and Monomerid = 50197263
TargetMetabotropic glutamate receptor 1(RAT)
Pfizer

Curated by ChEMBL
LigandPNGBDBM50197263((8-(4-methylpiperazin-1-yl)imidazo[1,2-a]pyrazin-2...)
Affinity DataKi:  1.09E+3nMAssay Description:Antagonist activity at rat mGluR1a expressed in CHO cells assessed as increase in calcium internalisation by FLIPR assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed