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Found 3 Enz. Inhib. hit(s) with Target = 'Glucocorticoid receptor' and Monomerid = 50197432
TargetGlucocorticoid receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50197432((4R)-4-[(1S,2S,5S,7R,9R,10R,11R,14R,16S)-9,16-dihy...)
Affinity DataKi:  4nMAssay Description:Displacement of radiolabeled Dexamethasone from human GRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50197432((4R)-4-[(1S,2S,5S,7R,9R,10R,11R,14R,16S)-9,16-dihy...)
Affinity DataKi:  15nMAssay Description:Inhibition of human GR expressed in hGRAF cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50197432((4R)-4-[(1S,2S,5S,7R,9R,10R,11R,14R,16S)-9,16-dihy...)
Affinity DataKi:  200nMAssay Description:Inhibition of human GR transcriptional activation by HepTAT cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed