Compile Data Set for Download or QSAR
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Found 3 Enz. Inhib. hit(s) with Target = 'Glucocorticoid receptor' and Monomerid = 50197434
TargetGlucocorticoid receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50197434(4-{[benzyl-(2-{[4-((9S,11R,13S,14S,17S)-17-hydroxy...)
Affinity DataKi:  1.10nMAssay Description:Displacement of radiolabeled Dexamethasone from human GRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50197434(4-{[benzyl-(2-{[4-((9S,11R,13S,14S,17S)-17-hydroxy...)
Affinity DataKi:  39nMAssay Description:Inhibition of human GR expressed in hGRAF cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50197434(4-{[benzyl-(2-{[4-((9S,11R,13S,14S,17S)-17-hydroxy...)
Affinity DataKi:  57nMAssay Description:Inhibition of human GR transcriptional activation by HepTAT cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed