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Found 2 Enz. Inhib. hit(s) with Target = 'Adenosine kinase' and Monomerid = 50201826
TargetAdenosine kinase(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50201826(6-(6-morpholin-4-ylpyridin-3-ylethynyl)-5-thiophen...)
Affinity DataIC50:  38nMAssay Description:Inhibition of cytosolic adenosine kinaseMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine kinase(Homo sapiens (Human))
Abbott Laboratories

Curated by ChEMBL
LigandPNGBDBM50201826(6-(6-morpholin-4-ylpyridin-3-ylethynyl)-5-thiophen...)
Affinity DataIC50:  212nMAssay Description:Inhibition of adenosine kinase in intact cells assessed as adenosine phosphorylationMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed