Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Glucocorticoid receptor' and Monomerid = 50216476
TargetGlucocorticoid receptor(Homo sapiens (Human))
Argenta Discovery

Curated by ChEMBL
LigandPNGBDBM50216476(5-(3-chlorobenzyl)-6-(4-benzylpiperidin-1-yl)-3-me...)
Affinity DataKi:  16nMAssay Description:Displacement of [3H]dexamethasone from human recombinant GRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Argenta Discovery

Curated by ChEMBL
LigandPNGBDBM50216476(5-(3-chlorobenzyl)-6-(4-benzylpiperidin-1-yl)-3-me...)
Affinity DataKi:  135nMAssay Description:Antagonist activity at human GRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed