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Found 2 Enz. Inhib. hit(s) with Target = 'Glucocorticoid receptor' and Monomerid = 50221156
TargetGlucocorticoid receptor(Homo sapiens (Human))
Corcept Therapeutics

Curated by ChEMBL
LigandPNGBDBM50221156(8a-(4-(piperidin-1-yl)benzyl)-2-(4-tert-butylpheny...)
Affinity DataKi:  9nMAssay Description:Displacement of [3H]dexamethasone from human glucocorticoid receptor expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Corcept Therapeutics

Curated by ChEMBL
LigandPNGBDBM50221156(8a-(4-(piperidin-1-yl)benzyl)-2-(4-tert-butylpheny...)
Affinity DataKi: >1.00E+3nMAssay Description:Antagonist activity at human glucocorticoid receptor in SW1353 cells assessed as inhibition of dexamethasone-induced luciferase expression by MMTV5 r...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed