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Found 4 Enz. Inhib. hit(s) with Target = 'Glucocorticoid receptor' and Monomerid = 50221173
TargetGlucocorticoid receptor(Homo sapiens (Human))
Corcept Therapeutics

Curated by ChEMBL
LigandPNGBDBM50221173((R)-8a-benzyl-2-(4-tert-butylphenylsulfonyl)-1,2,3...)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]dexamethasone from human recombinant GRMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Corcept Therapeutics

Curated by ChEMBL
LigandPNGBDBM50221173((R)-8a-benzyl-2-(4-tert-butylphenylsulfonyl)-1,2,3...)
Affinity DataKi:  4nMAssay Description:Displacement of [3H]dexamethasone from human glucocorticoid receptor expressed in recombinant baculovirusMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Corcept Therapeutics

Curated by ChEMBL
LigandPNGBDBM50221173((R)-8a-benzyl-2-(4-tert-butylphenylsulfonyl)-1,2,3...)
Affinity DataKi:  200nMAssay Description:Antagonist activity at GR in SW1353/MMTV5 cells assessed as inhibition of dexamethasone-induced luciferase expressionMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGlucocorticoid receptor(Homo sapiens (Human))
Corcept Therapeutics

Curated by ChEMBL
LigandPNGBDBM50221173((R)-8a-benzyl-2-(4-tert-butylphenylsulfonyl)-1,2,3...)
Affinity DataKi:  200nMAssay Description:Antagonist activity at human glucocorticoid receptor in SW1353 cells assessed as inhibition of dexamethasone-induced luciferase expression by MMTV5 r...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed