Compile Data Set for Download or QSAR
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Found 3 Enz. Inhib. hit(s) with Target = 'Gonadotropin-releasing hormone receptor' and Monomerid = 50225090
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50225090(CHEMBL399856 | isopropyl ((S)-2-(2-(1-(7-aza-bicyc...)
Affinity DataIC50:  3nMAssay Description:Antagonist activity at GnRH receptor expressed in AP Han Wistar rat primary pitutary cells assessed as inhibition of GnRH stimulated LH release after...More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Rattus norvegicus)
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50225090(CHEMBL399856 | isopropyl ((S)-2-(2-(1-(7-aza-bicyc...)
Affinity DataIC50:  15nMAssay Description:Displacement of [125I]D-Trp from rat GnRH receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetGonadotropin-releasing hormone receptor(Homo sapiens (Human))
Astrazeneca

Curated by ChEMBL
LigandPNGBDBM50225090(CHEMBL399856 | isopropyl ((S)-2-(2-(1-(7-aza-bicyc...)
Affinity DataIC50:  55nMAssay Description:Displacement of [125I]D-Trp from human GnRH receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed