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Found 5 Enz. Inhib. hit(s) with Target = 'Adenosine Receptor A2B' and Monomerid = 50229886
TargetAdenosine receptor A2b(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50229886(2-(3,4-Dimethoxy-phenyl)-N-[5-(2,6-dioxo-1,3-dipro...)
Affinity DataKi:  38nMAssay Description:Displacement of [3H]ZM241385 from human adenosine A2b receptor expressed in HEK cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50229886(2-(3,4-Dimethoxy-phenyl)-N-[5-(2,6-dioxo-1,3-dipro...)
Affinity DataKi:  38nMAssay Description:Binding affinity of compound for displacement of specific [3H]- DPCPX binding at human A2B receptors expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50229886(2-(3,4-Dimethoxy-phenyl)-N-[5-(2,6-dioxo-1,3-dipro...)
Affinity DataKi:  38nMAssay Description:Displacement of [3H]MRE2029F20 from human adenosine A2B receptor expressed in HEK293 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50229886(2-(3,4-Dimethoxy-phenyl)-N-[5-(2,6-dioxo-1,3-dipro...)
Affinity DataKi:  38nMAssay Description:Binding affinity of compound for displacement of [3H]DPCPX binding in HEK293 membranes expressing human A2B adenosine receptorsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
Cv Therapeutics

Curated by ChEMBL
LigandPNGBDBM50229886(2-(3,4-Dimethoxy-phenyl)-N-[5-(2,6-dioxo-1,3-dipro...)
Affinity DataIC50:  120nMAssay Description:Inhibitory activity against cAMP production in CHO cells transfected with human A2B adenosine receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed