Found 2 Enz. Inhib. hit(s) with Target = 'Muscarinic acetylcholine receptor M2' and Monomerid = 50231856
TargetMuscarinic acetylcholine receptor M2(Homo sapiens (Human))
Vanderbilt University Medical Center
Curated by ChEMBL
Vanderbilt University Medical Center
Curated by ChEMBL
Affinity DataIC50: >1.00E+4nMAssay Description:Antagonist activity at human muscarinic M2 receptor expressed in CHO-K1 cells coexpressing Gqi5 chimeric G-protein assessed as inhibition of acetylch...More data for this Ligand-Target Pair
TargetMuscarinic acetylcholine receptor M2(RAT)
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Vanderbilt Institute Of Chemical Biology
Curated by ChEMBL
Affinity DataIC50: >1.50E+5nMAssay Description:Antagonist activity at rat muscarinic M2 receptor expressed in CHO cells by calcium mobilization assayMore data for this Ligand-Target Pair