Compile Data Set for Download or QSAR
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Found 2 Enz. Inhib. hit(s) with Target = 'Progesterone receptor' and Monomerid = 50233022
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233022(2,2,2-trifluoro-N-((1S,13bR)-6-fluoro-1,3,4,13b-te...)
Affinity DataIC50:  730nMAssay Description:Inhibition of progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetProgesterone receptor(Homo sapiens (Human))
Nv Organon

Curated by ChEMBL
LigandPNGBDBM50233022(2,2,2-trifluoro-N-((1S,13bR)-6-fluoro-1,3,4,13b-te...)
Affinity DataEC50:  198nMAssay Description:Agonist activity at progesterone receptor expressed in CHO cells by luciferase assayMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed