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Found 2 Enz. Inhib. hit(s) with Target = 'Adenosine Receptor A2B' and Monomerid = 50233088
TargetAdenosine receptor A2b(Homo sapiens (Human))
East China University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50233088(1-ethyl-8-(1-(3-(trifluoromethyl)benzyl)-1H-pyrazo...)
Affinity DataKi:  6nMAssay Description:Antagonist activity against human adenosine A2B receptorMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetAdenosine receptor A2b(Homo sapiens (Human))
East China University Of Science And Technology

Curated by ChEMBL
LigandPNGBDBM50233088(1-ethyl-8-(1-(3-(trifluoromethyl)benzyl)-1H-pyrazo...)
Affinity DataKi:  6nMAssay Description:Displacement of [3H]-ZM241385 from human A2B receptor expressed in HEK293 cell membranesMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed