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Found 2 Enz. Inhib. hit(s) with Target = 'ATP-Binding Cassette Transporter ABCG2' and Monomerid = 50234479
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Universita Degli Studi Di Bari

Curated by ChEMBL
LigandPNGBDBM50234479(1,2-dimethoxy-4-((2-(3-methoxyphenethyl)phenoxy)me...)
Affinity DataIC50:  1.50E+5nMAssay Description:Inhibition of ABCG2 (unknown origin)More data for this Ligand-Target Pair
In DepthDetails ArticlePubMed
TargetBroad substrate specificity ATP-binding cassette transporter ABCG2(Homo sapiens (Human))
Universita Degli Studi Di Bari

Curated by ChEMBL
LigandPNGBDBM50234479(1,2-dimethoxy-4-((2-(3-methoxyphenethyl)phenoxy)me...)
Affinity DataEC50:  1.50E+5nMAssay Description:Inhibition of human BCRP pump mediated [3H]mitoxantrone transport in human Caco-2 cellsMore data for this Ligand-Target Pair
In DepthDetails ArticlePubMed